2
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T3072 | XL019 | Apoptosis , FLT , JAK , PDGFR | |
XL019 is a potent and selective JAK2 inhibitor with IC50 of 2.2 nM, 100 fold selectivity over JAK1. | |||
TQ0166 | Tesevatinib | KD-019,XL-647,EXEL-7647 | EGFR , VEGFR , FLT , Ephrin Receptor |
Tesevatinib (XL-647) is an orally available, multi-target tyrosine kinase inhibitor (IC50s: 0.3, 16, 1.5, 8.7, and 1.4 nM for EGFR, ErbB2, KDR, Flt4, and EphB4). |